What Is Sublingual Tirzepatide and How Does It Work?

What Is Sublingual Tirzepatide and How Does It Work?

About Tirzepatide

Tirzepatide is a medication that works on two important hormone pathways in the body: GLP-1 and GIP. These hormones affect appetite, digestion, and blood sugar control. By acting on both pathways, tirzepatide can support better glucose management and may help reduce hunger.

Sublingual Tirzepatide

In addition to injectable forms, tirzepatide may also be prescribed as a compounded sublingual formulation. This means the medication is absorbed through the tissue under the tongue, which allows it to enter the bloodstream directly. Sublingual formulations are not FDA-approved, but they can be prepared by licensed compounding pharmacies when prescribed by a healthcare provider.

Unlike injections, which are usually taken once weekly, sublingual tirzepatide drops are taken daily. Some patients may prefer this option because it offers a needle-free way to take the medication and allows for flexible dosing. Your provider will determine whether this approach is appropriate for you and guide you on how to use it properly.

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