About Tirzepatide
Tirzepatide is a medication that acts on hormone pathways involved in appetite and metabolism. Your healthcare provider may consider it as part of an individualized treatment plan based on your health needs.
Certain FDA-approved tirzepatide products have been studied in clinical trials for type 2 diabetes and weight management. Clinical studies of FDA-approved products apply only to those medications. Compounded formulations have not been evaluated by the FDA for safety or efficacy.
Sublingual Tirzepatide
Compounded sublingual tirzepatide is prepared by licensed compounding pharmacies when prescribed by a healthcare provider. These formulations are not FDA-approved and may differ from FDA-approved tirzepatide products in dosing, formulation, and available evidence.
Sublingual tirzepatide is taken by placing the prescribed amount under the tongue, following the instructions that accompany your prescription. Your provider will determine whether this type of formulation is appropriate for you.Administration timing and instructions may vary based on your prescription. Always follow the directions provided by your healthcare provider and the dispensing pharmacy.
Important Note
- Compounded sublingual tirzepatide is not FDA-approved.
- Your healthcare provider will determine whether this formulation is appropriate for you.
- Follow all administration instructions included with your prescription label or provided by your provider.

Compounded medications are not FDA-approved. They are prepared by licensed compounding pharmacies under medical supervision and may differ in formulation, dosing, and supporting evidence from FDA-approved products.

This article is for general informational purposes only and does not provide medical advice, diagnosis or treatment for any specific person.